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Barry, GD, Le, GT and Fairlie, DP (2006) Agonists and antagonists of protease activated receptors (PARs). Current Medicinal Chemistry, 13 3: 243-265. doi:10.2174/092986706775476070 214   43 Cited 44 times in Scopus44 0
Beyer, Renee L., Kelso, Michael J., Reid, Robert C., Le, Giang T. and Fairlie, David P. (2006). Alpha helix induction in HIV REV34-50 by N-terminal nucleators. In: Chemical Engineering News: Abstracts-232nd ACS National Meeting. 232nd ACS National Meeting, San Francisco, CA, U.S.A., (55-55). 10-14 September, 2006. doi:10.1021/cen-v084n034.p055 43   0
Iyer, Abishek, Fenning, Andrew, Lim, Junxian, Le, Giang T, Reid, Robert C, Halili, Maria A, Fairlie, David P and Brown, Lindsay (2010) Antifibrotic activity of an inhibitor of histone deacetylases in DOCA-salt hypertensive rats. British Journal of Pharmacology, 159 7: 1408-1417. doi:10.1111/j.1476-5381.2010.00637.x 137   34 Cited 43 times in Scopus43 0
Becker, B., Condie, G. C., Le, G. T. and Meutermans, W. (2006) Carbohydrate-based scaffolds in drug discovery. Mini-Reviews in Medicinal Chemistry, 6 12: 1299-1309. doi:10.2174/138955706778993003 94   15 Cited 15 times in Scopus15 0
Meutermans, Wim, Le, Giang Thanh and Becker, Bernd (2006) Carbohydrates as scaffolds in drug discovery. ChemMedChem, 1 11: 1164-1194. doi:10.1002/cmdc.200600150 23   85 Cited 87 times in Scopus87 0
Halili, Maria A., Ruiz-Gomez, Gloria, Le, Giang T., Abbenante, Giovanni and Fairlie, David P. (2009) Complement component C2, inhibiting a latent serine protease in the classical pathway of complement activation. Biochemistry, 48 35: 8466-8472. doi:10.1021/bi900679r 75   3 Cited 4 times in Scopus4 0
Halili, Maria A., Andrews, Melanie R., Labzin, Larisa I., Schroder, Kate, Matthias, Gabriele, Cao, Chun, Lovelace, Erica, Reid, Robert C., Le, Giang T., Hume, David A., Irvine, Katharine M., Matthias, Patrick, Fairlie, David P. and Sweet, Matthew J. (2010) Differential effects of selective HDAC inhibitors on macrophage inflammatory responses to the Toll-like receptor 4 agonist LPS. Journal of Leukocyte Biology, 87 6: 1103-1114. doi:10.1189/jlb.0509363 116   50 Cited 55 times in Scopus55 0
Cantley, M. D., Bartold, P. M., Marino, V., Fairlie, D. P., Le, G. T., Lucke, A. J. and Haynes, D. R. (2011) Histone deacetylase inhibitors and periodontal bone loss. Journal of Periodontal Research, 46 6: 697-703. doi:10.1111/j.1600-0765.2011.01392.x 37   8 Cited 8 times in Scopus8 0
Cantley, M. D., Fairlie, D. P., Bartold, P. M., Rainsford, K. D., Le, G. T., Lucke, A. J., Holding, C. A. and Haynes, D. R. (2011) Inhibitors of histone deacetylases in class I and class II suppress human osteoclasts in vitro. Journal of Cellular Physiology, 226 12: 3233-3241. doi:10.1002/jcp.22684 34   18 Cited 18 times in Scopus18 1
Suen, J. Y., Barry, G. D., Lohman, R. J., Halili, M. A., Cotterell, A. J., Le, G. T. and Fairlie, D. P. (2012) Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110). British Journal of Pharmacology, 165 5: 1413-1423. doi:10.1111/j.1476-5381.2011.01610.x 196   17 Cited 21 times in Scopus21 0
Loser, Reik, Abbenante, Giovanni, Madala, Praveen K., Halili, Maria, Le, Giang T. and Fairlie, David P. (2010) Noncovalent tripeptidyl benzyl- And cyclohexyl-amine inhibitors of the cysteine protease caspase-1. Journal of Medicinal Chemistry, 53 6: 2651-2655. doi:10.1021/jm901790w 40   4 Cited 5 times in Scopus5 0
Blakeney, J. S, Reid, R. C, Le, G. T and Fairlie, D. P (2007) Nonpeptidic ligands for peptide-activated G protein-coupled receptors. Chemical Reviews, 107 7: 2960-3041. doi:10.1021/cr050984g 89   57 Cited 55 times in Scopus55 0
Barry, Grant D., Suen, Jacky Y., Le, Giang T., Cotterell, Adam, Reid, Robert C. and Fairlie, David P. (2010) Novel agonists and antagonists for human protease activated receptor 2. Journal of Medicinal Chemistry, 53 20: 7428-7440. doi:10.1021/jm100984y 61   27 Cited 24 times in Scopus24 0
Yau, Annika M., Liu, Ligong, Reid, Robert C., Barry, Grant D., Suen, Jacky Y., Lohman, Rink-Jan, Le, Giang T., Cotterell, Adam and Fairlie, David P. (2011). Novel agonists and antagonists for protease activated receptor 2. In: Abstracts of Papers of the 242nd National Meeting of the American Chemical Society. National Meeting of the American Chemical Society (242nd, ACS, 2011), Denver, CO, U.S.A., (). 28 August-1 September 2011. 51   0
Le, G. T., Abbenante, G., Madala, P. K., Hoang, H. N. and Fairlie, D. P. (2006) Organic Azide Inhibitors of Cysteine Proteases. Journal of the American Chemical Society, 128 38: 12396-12397. doi:10.1021/ja0637649 82   11 Cited 12 times in Scopus12 0
Le, G. T, Abbenante, G. and Fairlie, D. P (2007) Profiling the enzymatic properties and inhibition of human complement factor B. Journal of Biological Chemistry, 282 48: 34809-34816. doi:10.1074/jbc.M705646200 70   11 Cited 10 times in Scopus10 0
Hoang, Huy N., Driver, Russell W., Beyer, Renée L., Malde, Alpeshkumar K., Le, Giang T., Abbenante, Giovanni, Mark, Alan E. and Fairlie, David P. (2011) Protein a-turns recreated in structurally stable small molecules. Angewandte Chemie International Edition, 123 47: 11303-11307. doi:10.1002/ange.201105119 72   6 Cited 6 times in Scopus6 0
Ruiz-Gomez, G, Lim, J, Halili, M. A., Le, G. T., Madala, P. K., Abbenante, G and Fairlie, D. P. (2009) Structure-activity relationships for substrate-based inhibitors of human complement factor B. JOURNAL OF MEDICINAL CHEMISTRY, 52 19: 6042-6052. doi:10.1021/jm900781m 57   4 Cited 4 times in Scopus4 0
Abbenante, G., Le, G. and Fairlie, D. P. (2007) Unexpected photolytic decomposition of alkyl azides under mild conditions. Chemical Communications, 2007 43: 4501-4503. doi:10.1039/b708134k 73   12 Cited 11 times in Scopus11 0