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Singh, Yogendra, Sharpe, Philip C., Hoang, Huy N., Lucke, Andrew J., McDowall, Alasdair W., Bottomley, Stephen P. and Fairlie, David P. (2011) Amyloid formation from an α-helical peptide bundle is seeded by 310-helix aggregates. Chemistry: A European Journal, 17 1: 151-160. doi:10.1002/chem.201002500 61   9 Cited 8 times in Scopus8 0
Sumanadasa, Subathdrage D. M., Goodman, Christopher D., Lucke, Andrew J., Skinner-Adams, Tina, Sahama, Ishani, Haque, Ashraful, Do, Tram Anh, McFadden, Geoffrey I., Fairlie, David P. and Andrews, Katherine T. (2012) Antimalarial activity of the anticancer histone deacetylase inhibitor SB939. Antimicrobial Agents and Chemotherapy, 56 7: 3849-3856. doi:10.1128/AAC.00030-12 69   17 Cited 15 times in Scopus15 1
Wheatley, Nicole C., Andrews, Katherine T., Tran, Truc L., Lucke, Andrew J., Reid, Robert C. and Fairlie, David P. (2010) Antimalarial histone deacetylase inhibitors containing cinnamate or NSAID components. Bioorganic & Medicinal Chemistry Letters, 20 23: 7080-7084. doi:10.1016/j.bmcl.2010.09.096 123   15 Cited 15 times in Scopus15 0
Xu, Weijun, Lucke A.J. and Fairlie D.P. (2015) Comparing sixteen scoring functions for predicting biological activities of ligands for protein targets. Journal of Molecular Graphics and Modelling, 57 76-88. doi:10.1016/j.jmgm.2015.01.009 36   0 Cited 0 times in Scopus0 3
Hill, Timothy A., Lohman, Rink-Jan, Hoang, Huy N., Nielsen, Daniel S., Scully, Conor C. G., Kok, W. Mei, Liu, Ligong, Lucke, Andrew J., Stoermer, Martin J., Schroeder, Christina I., Chaousis, Stephanie, Colless, Barbara, Bernhardt, Paul V., Edmonds, David J., Griffith, David A., Rotter, Charles J., Ruggeri, Roger B., Price, David A., Liras, Spiros, Craik, David J. and Fairlie, David P. (2014) Cyclic penta- and hexaleucine peptides without N-methylation are orally absorbed. ACS Medicinal Chemistry Letters, 5 10: 1148-1151. doi:10.1021/ml5002823 41   0 Cited 1 times in Scopus1 1
Lucke, AJ, Tyndall, JDA, Singh, Y and Fairlie, DP (2003) Designing supramolecular structures from models of cyclic peptide scaffolds with heterocyclic constraints. Journal of Molecular Graphics & Modelling, 21 5: 341-355. doi:10.1016/S1093-3263(02)00181-X 79   29 Cited 29 times in Scopus29 0
Kahnberg, P. C., Lucke, A., Glenn, M. P., Boyle, G. M., Tyndall, J. D., Parsons, P. G. and Fairlie, D. P. (2006) Design, Synthesis, Potency and Cytoselectivity of Anticancer Agents Derived by Parallel Synthesis from alpha-Aminosuberic Acid. Journal of Medicinal Chemistry, 49 26: 7611-7622. doi:10.1021/jm050214x 112   33 Cited 30 times in Scopus30 0
Lucke, Andrew J. and Young, David J. (2005) Electrophilic cleavage of cyclopropylmethystannanes: An experimental comparison of σ−σ and σ−π conjugation. Journal of Organic Chemistry, 70 9: 3579-3583. doi:10.1021/jo047822p 57   4 Cited 4 times in Scopus4 0
Cantley, M. D., Bartold, P. M., Marino, V., Fairlie, D. P., Le, G. T., Lucke, A. J. and Haynes, D. R. (2011) Histone deacetylase inhibitors and periodontal bone loss. Journal of Periodontal Research, 46 6: 697-703. doi:10.1111/j.1600-0765.2011.01392.x 43   11 Cited 11 times in Scopus11 0
Nielsen, Daniel S., Hoang, Huy N., Lohman, Rink-Jan, Hill, Timothy A., Lucke, Andrew J., Craik, David J., Edmonds, David J., Griffith, David A., Rotter, Charles J., Ruggeri, Roger B., Price, David A., Liras, Spiros and Fairlie, David P. (2014) Improving on nature: making a cyclic heptapeptide orally bioavailable. Angewandte Chemie - International Edition, 53 45: 12059-12063. doi:10.1002/anie.201405364 13   2 Cited 1 times in Scopus1 10
Cantley, M. D., Fairlie, D. P., Bartold, P. M., Rainsford, K. D., Le, G. T., Lucke, A. J., Holding, C. A. and Haynes, D. R. (2011) Inhibitors of histone deacetylases in class I and class II suppress human osteoclasts in vitro. Journal of Cellular Physiology, 226 12: 3233-3241. doi:10.1002/jcp.22684 38   20 Cited 19 times in Scopus19 1
Gupta, Praveer K., Reid, Robert C., Liu, Ligong, Lucke, Andrew J., Broomfield, Steve A., Andrews, Melanie R., Sweet, Matthew J. and Fairlie, David P. (2010) Inhibitors selective for HDAC6 in enzymes and cells. Bioorganic & Medicinal Chemistry Letters, 20 23: 7067-7070. doi:10.1016/j.bmcl.2010.09.100 65   14 Cited 13 times in Scopus13 0
Lucke, A., Boyle, G. M., Parsons, P. G. and Fairlie, D. (2006) New Cysteine Derivatives with Antiproliferative Activity on Melanoma Cells. Medicinal Chemistry, 2 2: 123-132. doi:10.2174/157340606776056124 57   2 Cited 2 times in Scopus2 0
Andrews, Kathy T., Tran, Thanh N., Lucke, Andrew, Kahnberg, Pia, Lee, G. T., Skinner-Adams, Tina, Gardiner, Donald L. and Fairlie, David P. (2007). Plasmodium falciparum histone deacetylases: Enzymes involved in gene regulation as new antimalarial drug targets. In: Abstract Book: American Society of Tropical Medicine and Hygiene : 56th Annual Meeting. 56th Annual Meeting of the American-Society-of-Tropical-Medicine-and-Hygiene, Philadelphia, PA United States, (48-48). 04-08 November 2007. 34   0
Andrews, K. T., Tran, T. N., Lucke, A. J., Kahnberg, P., Le, G. T., Boyle, G. M., Gardiner, D. L., Skinner-Adams, T. S. and Fairlie, D. P. (2008) Potent antimalarial activity of histone deacetylase inhibitor analogues. Antimicrobial agents and chemotherapy, 52 4: 1454-1461. doi:10.1128/AAC.00757-07 75   55 Cited 57 times in Scopus57 0
Singh, Y, Stoermer, MJ, Lucke, AJ, Glenn, MP and Fairlie, DP (2002) Regioselective synthesis of antiparallel loops on a macrocyclic scaffold constrained by oxazoles and thiazoles. Organic Letters, 4 20: 3367-3370. doi:10.1021/ol026463m 45   26 Cited 24 times in Scopus24 0
Singh, Y, Stoermer, MJ, Lucke, AJ, Guthrie, T and Fairlie, DP (2005) Structural mimicry of two cytochrome b(562) interhelical loops using macrocycles constrained by oxazoles and thiazoles. Journal of The American Chemical Society, 127 18: 6563-6572. doi:10.1021/ja0455300 70   28 Cited 29 times in Scopus29 0